Sr. No.ProductPharmacopoeiaDMF/CEP/WCTherapeutic Category
1Abiraterone AcetateIP / USP-NFODMFOral Hormone Therapy / Anti-cancer
2AcyclovirIP/ BP-EP / USP-NFODMFAntiviral
3Alpha Lipoic AcidIP/ BP-EP / USP-NFODMFNutritional / Antioxidant
4ApixabanIH / USP-NFODMFAnticoagulant
5ArtemetherIP / USP-NFODMF /WCAntimalarial
6Ascorbic Acid CoatedIHODMFNutritional / Vitamin
7BlonanserinIP/ BP-EP / USP-NFUnder preparationCNS (Antipsychotic)
8Bromfenac SodiumIP/ BP-EP / USP-NFUnder preparationOphthalmic / NSAID (Anti-inflammatory)
9CarbamazepineIP/ BP-EP / USP-NFODMFCNS (Anticonvulsant)
10DapagliflozinIP/ BP-EP / USP-NFODMFAntidiabetic (SGLT2 Inhibitor)
11Dapagliflozin Propanediol MonohydrateIP/ BP-EP / USP-NFUnder preparationAntidiabetic (SGLT2 Inhibitor)
12DeferasiroxPh. Eur.ODMFIron Chelator
13DihydroartemisininIHODMFAntimalarial
14EmpagliflozinIHODMFAntidiabetic (SGLT2 Inhibitor)
15FebuxostatIHODMFAnti-gout (Uric Acid Lowering)
16IlaprazoleIP / USP-NFUnder preparationA Proton Pump Inhibitor (PPI)
17IrbesartanIP/ BP-EP / USP-NFODMFAntihypertensive
18LevetiracetamIP/ BP-EP / USP-NFODMFAnti-convulsant
19LinezolidIP/ BP-EP / USP-NFODMFAnti-infective (Antibiotic)
20LumefantrineIP/ USP-NFODMF /WCAnti-infective (Antimalarial)
21MacitentanIHUnder preparationto treat Pulmonary Arterial Hypertension (PAH)
22MirogabalinIHUnder preparationCNS (Neuropathic Pain)
23NorfloxacinIP/ BP-EP / USP-NFODMFAnti-infective (Fluoroquinolone)
24OfloxacinIP/ BP-EP / USP-NFODMF /WCAnti-infective (Fluoroquinolone)
25OxcarbazepineIP/ BP-EP / USP-NFODMFCNS (Anticonvulsant)
26Oxymetazoline HydrochlorideIP/ BP-EP / USP-NFODMFTopical / ENT (Decongestant)
27PolmacoxibIHUnder preparationNSAID
28PregabalinIP/ BP-EP / USP-NFODMFCNS (Neuropathic Pain / Anticonvulsant)
29PrilocaineIP/ BP-EP / USP-NFODMFTopical / Local Anesthetic
30RivaroxabanIP/ BP-EP / USP-NFODMFCardiovascular (Anticoagulant)
31RivaroxabanIHODMFAnticoagulant
32Tamsulosin HydrochlorideIP/ BP-EP / USP-NFODMFUrology (BPH / Alpha Blocker)
33ValacyclovirIP/ BP-EP / USP-NFUnder preparationAntiviral
34ValganciclovirIP/ BP-EP / USP-NFUnder preparationAntiviral
35Xylometazoline HydrochlorideIP/ BP-EP / USP-NFODMFTopical / ENT (Decongestant)
Sr. No. Product Name Intermidiate Name CAS NO
1diltiazimCIS (+) Hydroxy Lactum42399-49-5
2perxitine(-)4-(4-Fluorophenyl)-3-Hydroxy methyl-1-methyl Piperidine105812-81-5
3vildagliptin3-Amino-1-Adamantan 702-82-9
4oxcarbamezipine10-methoxy iminostilbine 4698.-11-7
5triptilin3-Dimethylaminopropylchloride hydrochloride5407-04-5.
6Amiodarone HCL Amiodarone HCL 1951-25-3
7APIXABAN1-(4-IODO-PHENYL)-PIPERIDIN-2-ONE385425-15-01-(4-BROMO-PHENYL)-PIPERIDIN-2-ONE27471-43-81-( 4-NITRO-PHENYL)-PIPERIDIN-2-ONE38560-30-4ETHYL CHLORO[(4-METHOXYPHENYL)HYDRAZONO]ACETATE27143-07-3/473927-63-82-PIPERIDONE675-20-73-CHLORO-5,6-DIHYDRO-1-(4-NITROPHENYL)-2(1H)-PYRIDINONE536760-29-93-MORPHOLIN-4-YL-1-(4-NITROPHENYL)-5,6-DIHYDROPYRIDIN-2(1H)-ONE503615-03-0ETHYL 1-(4-METHOXYPHENYL)-6-(4-NITROPHENYL)-7-OXO-4,5,6, 7-TETRAHYDRO-1H-PYRAZOLO[3,4-C]PYRIDINE-3-CARBOXYLATE536759-91-81-(4-IODOPHENYL)-3-MORPHOLINE-4-YL-5,6DIHYDROPYRIDINE-2 ONE473927-69-4ETHYL- 1-(4-METHOXYPHENYL)-7-OXO-6-[4-(2-OXOPIPERIDIN-1-YL) PHENYL]-4,5-DIHYDROPYRAZOLO[5,4-C]PYRIDINE-3-CARBOXYLATE503614-91-33-MORPHOLINO-1-[4-(2-OXOPIPERIDIN-1-YL)PHENYL]-5,6- DIHYDROPYRIDIN-2(1H)-ONE545445-44-13,3-DICHLORO-1-(4-NITROPHENYL)PIPERIDIN-2-ONE881386-01-21(4-AMINOPHENYL)-3-MORPHOLIN-4YL-5,6 DIHYDROPYRIDINE-2(1H)-ONE1267610-26-3ETHYL 1-(4-METHOXYPHENYL)-6-(4-IODOPHENYL)-7-OXO-4,5,6,7- TETRAHYDRO-1H-PYRAZOLO[3,4-C]PYRIDINE-3-CARBOXYLATE473927-64-9
8APREMILAST3-NITRO PHTHALIC ACID603-11-23-AMINO PHTHALIC ACID5434-20-83-ETHOXY-4-METHOXY BENZALDEHYDE1131-52-83-ETHOXY-4-METHOXY BENZONITRILE60758-86-33-ACETAMIDO PHTHALIC ANHYDRIDE6296-53-3
9ARIPIPRAZOLE1-(2,3-DICHLORO PHENYL) PIPERAZINE HCl119532-26-2
10CABOZANTINIB6,7-DIMETHOXYQUINOLIN-4-OL13425-93-94-CHLORO-6,7-DIMETHOXYQUINOLINE35654-56-9CYCLOPROPANE-1,1-DICARBOXYLIC ACID598-10-71-((4-FLUOROPHENYL)CARBAMOYL)CYCLOPROPANE-1-CARBOXYLIC ACID849217-48-74-((6,7-DIMETHOXY-QUINOLIN-4-YL)OXY)ANILINE190728-25-74-[(6,7-DIMETHOXYQUINOLIN-4-YL)OXY]ANILINE] ACID190728-24-6
11CARBOPLATIN1-(CYCLOPROPYLCARBONYL)PIPERAZINE HYDROCHLORIDE1021298-67-81,1-CYCLOBUTANE DICARBOXYLICACID5445-51-2
12CELECOXIB4-HYDRAZINOBENZENESULFONAMIDE27918-19-0
13CILOSTAZOL6-HYDROXYL-3,4-DIHYDRO-2(1H)-QUINOLINONE54197-66-9
14CLOFAZAMINEN-(4-CHLOROPHENYL)2-NITROANILINE23008-56-2
15DABIGATRAN4-(METHYLAMINO)-3-NITROBENZOIC ACID41263-74-5ETHYL -3- (PYRIDINE-2YL AMINO ) PROPANOATE103041-38-9ETHYL 3-[{3-AMINO-4-(METHYL AMINO)BENZOYL}(PYRIDIN-2-YL)AMINO]-PROPANOATE212322-56-04-CHLORO-3-NITROBENZOIC ACID96-99-14-CYNO PHENYL GLYCINE42288-26-6
16DOLUTEGRAVIRAMINOACETALDEHYDE DIMETHYL ACETAL23008-56-21-(2,2-DIMETHOXYETHYL)-5-METHOXY-6-(METHOXYCARBONYL) -4-OXO-1,4-DIHYDROPYRIDINE-3-CARBOXYLIC ACID41263-74-5METHYL-4-METHOXY ACETOACETAE103041-38-9
17DOLUTEGRAVIR/IMATINIBN,N-DIMETHYL FORMAMIDE DIMETHYL ACETAL4637-24-5
18EDOXABAN5-METHYL-4,5,6,7-TETRAHYDROTHIAZOLO [5,4-C]PYRIDINE-2-CARBOXYLIC ACID HCL720720-96-72-AMINO-5-METHYL-4,5,6,7-TETRAHYDROTHIAZOLO[5,4-C]PYRIDINE17899-48-85-METHYL-4,5,6,7-TETRAHYDROTHIAZOLE[5,4-C]PYRIDINE TOSYLATE259809-24-02-BROMO-5-METHYL-4,5,6,7-TETRAHYDROTHIAZOLO[5,4-C]PYRIDINE TOSYLATE143150-92-92-[(5-CHLOROPYRIDIN-2-YL)AMINO]-2-OXOACETIC ACID ETHYL ESTER HCI1243308-37-3
19ELTROMBOPAG3,4-DIMETHYLPHENYLHYDRAZINE HCl60481-51-82-BROMO-6-NITROPHENOL13073-25-12-(3,4-DIMETHYLPHENYL)-5-METHYL-2,4-DIHYDRO-3H-PYRAZOL-3- ONE277299-70-4
20ETODOLAC7-ETHYL TRYPTOPHOL41340-36-7
21FORETINBCYCLOPROPANE-1 1-DICARBOXYLIC ACID598-10-7
22HOMOTAURINE3-AMINO-1-PROPANE SULPHONIC ACID3687-18-1
23LABETALOL5-(N,N-DIBENZYLGLYCYL)SALICYLAMIDE30566-92-85-BROMOACETYL-SALICYLAMIDE73866-23-65-CHLOROACETYL-SALICYLAMIDE5-(CHLOROACETYL)-2-HYDROXYBENZAMIDE33254-88-5
24LOSARTANVALERONITRILE110-59-8
25MACITENTANDIMETHYL(4-BROMOPHENYL)MALONATE14906-35-45-(4-BROMOPHENYL)PYRIMIDINE-4,6-DIOL706811-25-85-(4-BROMOPHENYL)-4,6-DICHLOROPYRIMIDINE146533-41-75-BROMO-2-CHLOROPYRIMIDINE32779-36-5
26MECARBINATEETHYL 5-HYDROXY-1,2-DIMETHYL-1H-INDOLE-3-CARBOXYLATE15574-49-9
27NINTEDANIBTRI METHYL ORTHO BENZOATE707-07-3TRI ETHYL ORTHO BENZOATE1663-61-2METHYL-4-CHLORO-3-NITRO BENZOIC ACID14719-83-6N-METHYL-4-NITROANILINE100-15-2
28NINTEDANIB2-CHLORO-N-METHYL-N-(4-NITROPHENYL) ACETAMIDE2653-16-9N-METHYL-2-(4-METHYLPIPERAZIN-1-YL)-N-(4-NITROPHENYL) ACETAMIDE1139453-98-7N-METHYL-2-(4-METHYLPIPERAZIN-1-YL)-N-(4-AMINOPHENYL) ACETAMIDE262368-30-9METHYL 1-ACETYL-2-OXOINDOLINE-6-CARBOXYLATE676326-36-61,3-DIMETHYL 2-[4-(METHOXYCARBONYL)-2-NITROPHENYL]PROPANEDIOATE1160293-27-56-METHOXYCARBONYL-2-OXINDOLE14192-26-84-CHLORO-3-NITROBENZOIC ACID96-99-12-BROMO-N-METHYL-N-(4-NITROPHENYL)ACETAMIDE23543-31-9
29ORMELOXIFENE1-(2-HYDROXY ETHYL)PYRROLIDINE2955-88-6
30PAZOPANIB5-AMINO-2-METHYLBENZENESULFONAMIDE6973-09-72,4-DICHLORO PYRIMIDINE3934-20-1
31PENTOXIFYLLINE6-CHLORO 2-HEXANONE10226-30-9
32PIMAVANSERIN4-ISOBUTOXY BENZYLAMINE HCl SALT37806-44-34-ISOBUTOXY BENZYLAMINE ACETATE955997-89-44-ISOBUTOXY BENZALDEHYDE18962-07-7
33POSACONAZOLE1-(4-HYDROXYPHENYL)PIPERAZINE56621-48-81-(4-HYDROXYPHENYL)-4-(4-AMINO PHENYL)PIPERAZINE74853-08-0
34QUETIAPINE1-[2-(2-HYDROXY ETHOXY)ETHYL]PIPERAZINE13349-82-1DIBENZO[B,F][1,4]THIAZEPIN-11(10H)-ONE3159-07-7
35RANOLAZINEGUAIACOL GLYCIDYL ETHER2210-74-4N-(2,6-DIMETHYLPHENYL)-2-(PIPERAZIN-1-YL)ACETAMIDE5294-61-1
36RIBOCICLIB/ PALBOCICLIB5-BROMO -2-NITRO PYRIDINE39856-50-36-BROMO-2-CHLORO-8-CYCLOPENTYL-5-METHYLPYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE1016636-76-25-BROMO-2-CHLORO-N-CYCLOPENTYLPYRIMIDIN-4-AMINE733039-20-85-BROMO-2,4-DICHLOROPYRIMIDINE36082-50-51-BOC- 4-(6-NITRO-3-PYRIDYL)PIPERAZINE571189-16-71-BOC- 4-(6-AMINO-3-PYRIDYL)PIPERAZINE571188-59-5
37RIVAROXABAN2-[[(5S)-2-OXO-3-[4-(3-OXO-4-MORPHOLINYL)PHENYL]-5-OXAZOLIDINYL]METHYL]-1H- ISOINDOLE-1,3(2H)-DIONE446292-08-64-(4-NITROPHENYL)MORPHOLIN-3-ONE446292-04-24-(4-AMINOPHENYL)MORPHOLIN-3-ONE438056-69-0S-(2,3-EPOXYPROPYL)PHTHALAMIDE161596-47-0
38SITAGLIPTINMELDRUM'S ACID2033-24-1
39TRAZODONE2H-[1,2,4]TRIAZOLO[4,3-A]PYRIDINE-3-ONE6969-71-71-(3-CHLOROPHENYL)-4-(3-CHLOROPROPYL)PIPERAZINE HCL52605-52-41-(3 CHLORO PHENYL)PIPERAZINE6640-24-01-(3 CHLORO PHENYL)PIPERAZINE HCL65369-76-8 /13078-15-4
40VELBANAZINE(N,N-DIMETHYL AMINO METHYL)-5-METHYL-2-HEXANONE OXALATE SALT2102090-17-33, 4- DIHYDRO-6, 7- DIMETHOXY-ISOQUINOLINE3382-18-13,4-DIHYDRO-6,7-DIMETHOXY-ISOQUINOLINE HYDROCHLORIDE20232-39-7
41VILAZODONEETHYL-5-PIPRAZINYL BENZOFURAN-2-CARBOXYLATE HCL765935-67-9ETHYL-5-NITROBENZOFURAN-2-CARBOXYLATE69604-00-8ETHYL-5-AMINO BENZOFURAN-2-CARBOXYLATE174775-48-55-AMINOBENZOFURAN-2-CARBOXYLIC ACID42933-44-85-PIPERAZINEYL-BENZOFURAN-2CARBOXAMIDE183288-46-2N,N-BIS(2-CHLOROETHYL)-4-METHYLBENZENE SULFONAMIDE42137-88-2
42VILDAGLIPTIN3-HYDROXY-1-ADAMANTAN AMINE702-82-9
43VORTIOXETINE2,4-DIMETHYL THIOPHENOL13616-82-5N-BOC-PIPERAZINE57260-71-6
44ZIPRASIDONE1-(1,2-BENZISOTHIAZOL-3-YL) PIPERAZINE87691-87-0
45ZONISAMIDESODIUM BENZO[D]ISOXAZOL-3-YL-METHYLSULFONATE73101-64-1
46ZONISAMIDE/ WARFRAIN4-HYDROXY COUMARINE1076-38-6
47
47
50ACOTIAMIDEN,N-DIISOPROPYLETHYLENE DIAMINE121-05-1
51BEMPEDOIC ACIDETHYL-2,2-DIMETHYL-7-BROMOHEPTANOATE123469-92-1P-TOLUENESULFONYLMETHYL ISOCYANIDE36635-61-7
52BORTEZOMIBN-(2-PYRAZINE CARBONYL)-L-PHENYL ALANINE114457-94-2
53BREXPIPRAZOLE7-HYDROXYQUINOLIN-2(1H)-ONE70500-72-0N-(CINNAMOYL)-3-METHOXYANILINE127033-74-34-CHLORO-1-BENZOTHIOPHENE-2-CARBOXILIC ACID23967-57-94-CHLORO-1-BENZOTHIOPHENE66490-33-31-(1-BENZOTHIOPHEN-4-YL)PIPERAZINE HCl913614-18-3
54BUTORPHANOLCYCLOBUTANE CARBOXYLIC ACID3721-95-7
55CARFILZOMIBMORPHOLINE ACETIC ACID HCl3235-69-6
56CERITINIB / BRIGATINIB2,4,5-TRICHLOROPYRMIDINE5750-76-5
57CETIRIZINE2-(2-CHLORO ETHOXY) ETHYL ACETATE14258-40-3
58CIZOLIRTIN1-METHYL-1H-PYRAZOLE930-36-9
59CLOFAZAMINE2-AMINO-4-CHLORO DIPHENYLAMINE68817-71-0
60CRIZOTINIB4-IODO PYRAZOLE3469-69-0
61EFINACONAZOLE4-METHYLENE PIPERIDINEHYDROCHLORIDE144230-50-2
62ERLOTINIBETHYL-2-AMINO-4,5-BIS-(2-METHOXYETHOXY) BENZOATE HCl183322-17-06,7-BIS-(2-METHOXYETHOXY)-4(3H)-QUINAZOLINONE179688-29-0
63FALNIDAMOL1-METHYLPIPERIDIN-4-AMINE41838-46-4
64FEDRATINIB1-(2-CHLOROETHYL)PYRROLIDINE7520-67-13-AMINO-N-(TERT-BUTYL)BENZENESULPHONAMIDE608523-94-0
65FLIBANSERIN1,3-DIHYDRO-2H-BENZIMIDAZOLE-2-ONE615-16-71-ISOPROPENYL-2-BENZIMIDAZOLIDINONE52099-72-61-(2-CHLOROETHYL)-1,3-DIHYDRO-2H-BENZIMIDAZOL-2-ONE52548-84-21-(2-BROMOETHYL)-1,3-DIHYDRO-2H-BENZIMIDAZOL-2-ONE103784-03-81-[3-(TRIFLUOROMETHYL)PHENYL]PIPERAZINE HCl76835-14-84-[3-TRIFLUOROMETHYL)PHENYL]-1-(2-CHLOROETHYL) PIPERAZINEDIHYDROCHLORIDE57061-71-9
66FLORDIPINE4-(2-AMINO ETHYL) MORPHOLINE2038-03-1
67HYDROCHLOROTHIAZIDE5-CHLORO-2,4-DISULFAMOYLANILINE
68LETERMOVIR1-(3-METHOXYPHENYL) PIPERAZINE16015-71-7
69LOMITAPIDE4-(N-BOC-AMINO) PIPERIDINE73874-95-04-AMINO-N-BENZYL PIPERIDINE50541-93-0
70LULICONAZOLE1H-IMIDAZOL-1-YLACETONITRILE HYDROCHLORIDE98873-55-31-(CYANO METHYL) IMIDAZOLE HYDROCHLORIDE]220476-15-32-BROMO-1-(2,4-DICHLOROPHENYL)ETHANONE2631-72-3
71
72LUMATAPERONEETHYL (6BR,10AS)-METHYL-2,3,6B,9,10,10A-HEXAHYDRO-1H- PYRIDO[3',4'4,5]PYRROLO[1,2,3-DE]QUINOXALINE-8(7H)-CARBOXYLATE313369-26-52-BROMOPHENYLHYDRAZINE HYDROCHLORIDE50709-33-62-CHLORO-N-METHYLACETAMIDE96-30-04-PIPERIDONE MONOHYDRATE HYDROCHLORIDE40064-34-4N,N-DIMETHYL ETHYLENE DIAMINE110-70-3
73METYROSINE4-BROMOPHENETOLE588-96-5N-METHYL-2,4-DINITRO ANILINE2044-88-4
74MILICICLIB1-(4-AMINOPHENYL)-4-METHYLPIPERAZINE16153-81-4ETHYL (HYDROXYIMINO)CYANOACETATE3849-21-6
75NAFTOPIDILE / URAPIDIL1-(2-METHOXY PHENYL)PIPERAZINE HCl5464-78-8
76OLAPARIBCYCLOPROPYL CARBONYL PIPERAZINE59878-57-8
77OSPEMIFENE2-(4-BROMOPHENOXY)TATRAHYDROPYRAN36603-49-3BENZYL-2-BROMOETHYLETHER1462-37-92-(2-BROMOETHOXY)TETRAHYDROPYRAN17739-45-6
78POMALIDOMIDE3-NITROPHTHALIC ANHYDRIDE641-70-3
79PROPRANOLOL2-[(1-NAPHTHYLOXY)METHYL]OXIRANE2461-42-9
80PRUCALOPRIDE1-CHLORO-3-METHOXYPROPANE36215-07-31-(3-METHOXYPROPYL)PIPERIDIN-4-ONE16771-85-01-(3-METHOXYPROPYL)PIPERIDIN-4-AMINE179474-79-44-(N-BOC AMINO) PIPERIDINE73874-95-0
81REGORAFENIB4-CHLORO-N-METHYLPYRIDINE-2-CARBOXAMIDE HCL882167-77-34-(4-AMINO-3-FLUOROPHENOXY)-N-METHYLPYRIDINE-2-CARBOXAMIDE757251-39-1
81REPAGLINIDEN-ACETYL-L-GLUTAMICACID1188-37-0
83RILPIVIRINE4-IODO-2,6-DIMETHYLANILINE4102-53-8
84ROFLUMILAST4-AMINO-3,5-DICHLOROPYRIDINE22889-78-7
85SACUBITRILETHYL-2-(TRIPHENYLPHOSPHORANYLIEDINE)PROPANOATE5717-37-3
86SATAVAPTAN4-(2-CHLORO ETHL)MORPHOLINE3240-94-6
87SELEXIPAG5,6-DIPHENYLPYRAZIN-2-OL18591-57-64-(ISOPROPYL AMINO)BUTANOL42042-71-7METHANE SULPHONAMIDE3144-09-05-BROMO-2,3-DIPHENYLPYRAZINE243472-70-0
88SORAFENIB4-(4-AMINOPHENOXY)-N-METHYLPYRIDINE-2-CARBOXAMIDE284462-37-9
89SUVOREXANTN-BOC-ETHYLENE DIAMINE57260-73-8
90TIOTROPIUM BROMIDEMETHYL-2,2-DITHIENYL GLYCOLATE26447-85-8
91VOLSARTIB3-METHOXY-4-NITRO BENZOIC ACID5081-36-7CYCLOPROPYL METHYL PIPERAZINE57184-25-5
923-PHENYLMETHYL)AMINO-1-PROPANOL4720-29-0
931-BOC-4-PIPERIDONE79009-07-3
94(2-BROMOETHYL)BENZENE103-63-9
951-BENZYL-4-(4-FLUOROPHENYL)PIPERIDIN-4-OL163631-02-5
961-BOC-4-(HYDROXYMETHYL)-PIPERIDINE123855-51-6
971-BROMO-6(TRIMETHYLAMMONIUM)HEXYL BROMIDE32765-81-4
981-ISOPROPYL-1H-PYRAZOLE18952-87-9
991-METHANESULFONYLPIPERAZINE HCl55276-43-2
1002,3-DIHYDRO-2-OXO-1H-BENZIMIDAZOLE-1-BUTYRIC ACID (BUZOLIC ACID)3273-68-5
1012,4-DICHLORO-6,7-DIHYDROTHIENO[3,2-D]PYRIMIDINE74901-69-2
1022,5-BIS-ACETAMIDO-3,6-DICHLORO-BENZOQUINONE10541-83-0
1032-BROMO BENZONITRILE2042-37-7
1042-BROMO-4-FLUOROACETOPHENONE403-29-2
1052-CHLORO-1,1,1-TRIETHOXYETHANE51076-95-0
1062-ISOPENTYL-2-ISOPROPYL-1,3-DIMETHOXYPROPANE129228-11-1
964-(4-FLUOROPHENYL)PIPERIDIN-4-OL3888-65-1
974-AMINO-N-TERT-BUTYLBENZENESULFONAMIDE209917-48-6
984-BROMO-1-METHYL-1H-PYRAZOLE15803-02-8
995,6-DIAMINO-1,3-DIHYDRO-2H-BENZIMIDAZOL-2-ONE55621-49-3
100BENZYL HYDRAZINE DIHYDROCHLORIDE20570-96-1
101CYCLOBUTYL PIPERAZINE61379-68-8
102ISOPROPYL MYRISTATE110-27-0
103N,N-DIMETHYL FORMAMIDE DITERT BUTYL ACETAL36805-97-7
104N-AMINOPHTHALIMIDE1875-48-5
105N-BUTYL PIPERAZINE5610-49-1
106N-ETHYLBENZYLAMINE14321-27-8
107N-METHYL-2-CYANOACETAMIDE6330-25-2
108CHLORO ACETONITRILE107-14-2
109GLYCINE METHYL ESTER HYDROCHLORIDE5680-79-5
110AMLODIPINEN-(2-HYDROXYETHYL)PHTHALIMIDE3891-07-4N-(2-CHLOROETHYL)PHTHALIMIDE6270-06-0
111BAZEDOXIFENE4-BENZYLOXYPROPIOPHENONE4495-66-31-(BENZYLOXY)-4-NITROBENZENE1145-76-24-(BENZYLOXY)-ANILINE HCL51388-20-6
112BETRIXABAN2-AMINO-5-CHLOROPYRIDINE1072-98-6N-(5-CHLOROPYRIDIN-2-YL)-5-METHOXY-2-NITROBENZAMIDE280773-16-22-AMINO-N-(5-CHLOROPYRIDIN-2-YL)-5-METHOXYBENZAMIDE280773-17-3N-(5-CHLOROPYRIDIN-2-YL)-2-[(4-CYANOBENZOYL)AMINO]-5-METHOXYBENZAMIDE330942-01-3
113BILASTINE2-(PIPERIDIN-4-YL)-1H—BENZIMIDAZOLE38385-95-4
114BRIGATINIB2-METHOXY-4-[4-(4-METHYLPIPERAZIN-1-YL)PIPERIDIN-1-YL]ANILINE761440-25-91-METHYL-4-(PIPERIDIN-4-YL)-PIPERAZINE53617-36-0
115BUSPIRONEN-(2-PYRIMIDINYL)-PIPERAZINE20980-22-7
116DEUCRAVACITINIBCYCLOPROPANE CARBOXAMIDE6228-73-52-METHOXY-3-NITROBENZONITRILE121001-06-7N-METHYL-N-FORMYLHYDRAZINE758-17-8
117OPICAPONE3,4-DIMETHOXY-5-NITROBENZALDEHYDE22027-96-9
118OSIMERTINIB3-(2-CHLOROPYRIMIDIN-4-YL)-1-METHYLINDOLE1032452-86-0N,N,N'-TRIMETHYL ETHYLENE DIAMINE142-25-6
119PONATINIB4-(4-METHYL-PIPERAZIN-1-YLMETHYL)-3-TRIFLUORO METHYL PHENYLAMINE694499-26-8
120PYRANTEL & OXANTEL1,2-DIMETHYL-1,4,5,6-TETRAHYDROPYRIMIDINE4271-96-9
121REVEFENACINBENZYL METHYL-(2-OXOETHYL)CARBAMATE107201-33-2
122RILPIVIRINE4-[(4-CHLORO-2-PYRIMIDINYL) AMINO BENZONITRILE244768-32-9
123SUNITINIBN-[2-(DIETHYLAMINO)ETHYL]-3-OXOBUTANAMIDE590424-03-6
124TIROFIBAN1-BOC-4-(2-HYDROXYETHYL)PIPERIDINE89151-44-0
125TRILACICLIB5-(4-METHYLPIPERAZIN-1-YL)PYRIDIN-2-AMINE571189-49-6
126Alogliptin(R)-3-Amino-piperidine dihydrochloride334618-23-4
127Linagliptin
128Trelagliptin
129Alogliptin(R)-3-(Boc-Amino)piperidine309956-78-3
130Linagliptin
131Trelagliptin
132BendamustineEthyl 4-(1-methyl-5-nitro-1H-benzo[d] imidazol-2-yl)butanoate3543-72-4
133BendamustineEthyl4-(5-amino-1-methyl-1H-benzo[d]imidazole -2-yl)butanoate3543-73-5
134Cabozantinib4-chloro-6,7-dimethoxyquinoline35654-56-9
135Camostat mesylate4- Guanidinobenzoic Acid HCl42823-46-1
136Camostat mesylate2-Chloro-N,N-dimethylacetamide2675-89-0
137Camostat mesylate4-Hydroxy Benzeneacetic Acid2-(Dimethylamino)-2-oxoethyl Ester59721-16-3
138Cinacalcet3-(3-Trifluoromethylphenyl)propionic Acid585-50-2
139Cinacalcet(R)-N-(1-(naphthalen-1-yl)ethyl)-3-(3-(trifluoromethyl)phenyl)propanamide1005450-55-4
140Droxidopa3,4-Dibenzyloxybenzaldehyde09-02-5447
141DabigatranEthyl 3(-4-(ethyl amino)-3- nitro-N-(pyridin-2-yl)benzamido)propanoate429659-01-8
142DabigatranEthyl 3-(3-amino-4-(methyl amino)-N-(pyridin-2-yl) benzamido) propanoate212322-56-0
143Dabigatran2-(4-Cyanophenylamino) Acetic Acid42288-26-6
144DabigatranEthyl-3-[[[2-[[(4-cyanophenyl) amino] methyl]-1methyl-1H-benzimidazol-5-yl]carbonyl]pyridine-2-ylamino] propionate.211915-84-3
145DabigatranEthyl 3-(2-(((4-carbamimidoylphenyl)amino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanoate hydrochloride.211914-50-0
146Dasatinib2-(N-BOC)-Aminothiazole-5-carboxylic acid302964-02-9
147Dasatinib(E) -N-(2-Chloro-6-Methyl Phenyl)-3-Ethoxy Acrylamide863127-76-8
148Dasatinib2-Amino-N-(2-chloro-6-methylphenyl)thiazole-5-carboxamide302964-24-5
149Dasatinib4,6-dichloro-2-methylpyrimidine1780-26-3
150ElagolixN-Boc-D-phenyl glycinol102089-74-7
151Elagolix(R)-2-(tert-butoxycarbonylamino)-2-phenylethyl methanesulfonate102089-75-8
152Eliglustat2,3-dihydrobenzo[b][1,4]dioxine-6-carbaldehyde29668-44-8
153EliglustatS(+)-2-Phenylglycinol20989-17-7
154Ibandronate3-(N-Methyl-N-Pentyl amino)propionic acid HCl625120-81-2
155Icotinib(ethane-1,2-diylbis(oxy)) bis(ethane-2,1-diyl) bis(4-methylbenzenesulfonate)19249-03-7
156Icotinib2-amino-4,5-dimethoxybenzoic acid5653-40-7
157Imatinib4-[(4-Methylpiperazin-1-yl)-methyl]-benzoic acid dihydrochloride106261-49-8
158ImatinibN-(5-Amino-2-methylphenyl)-4-(3-pyridyl)-2-pyrimidineamine152460-10-1
160Ibrutinib4-Aminopyrazolo[3,4-d]pyrimidine2380-63-4
161Ibrutinib3-(4-Phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine330786-24-8
162Ivacaftor4-oxo-1,4-dihydroquinoline-3-carboxylic acid (USDMF No. 33616)13721-01-2
163IvacaftorEthyl 4-Oxo-1,4-dihydroquinoline-3-carboxylate52980-28-6
164Ivacaftor5-Amino-2,4-ditert-butylphenol873055-58-4
165Ivacaftor5-Amino-2,4-ditert-butylphenol hydrochloride1777786-05-6
166Mirabegron2-(2-Aminothiazol-4-yl)acetic acid29676-71-9
167Mirabegron2-(2-Aminothiazol-4-yl)acetic acid hydrochloride66659-20-9
168Mirabegron2-(4-nitrophenyl)ethanamine hydrochloride29968-78-3
169Mirabegron(R)-2-(4-nitrophenethylamino)-1-phenylethanol hydrochloride521284-21-9
170MirabegronR)-2-(4-nitrophenethylamino)-1- Phenylethanol (USDMF No. 35841)223673-34-5
171Mirabegron(R)-2-(4-aminophenethylamino)-1-Phenylethanol hydrochloride521284-22-0
172Mirabegron(R)-2-((4-Aminophenethyl)amino)-1-phenylethanol391901-45-5
173MolnupiravirN-Hydroxycytidine acetonide ester2346620-55-9
174Ondansetron1,2,3,9-tetrahydro-9-methyl-4H-carbazol-4-one27387-31-1
175Ondansetron3-[(Dimethylamino)methyl]-1,2,3,9-tetrahydro-9-methyl-4H-carbazol-4-one HCl119812-29-2
176Paliperidone4-(6-Fluoro-1,2-benzisoxazole-3yl)-Piperidine Hydrochloride84163-13-3
177Risperidone
178Paliperidone4-[2,4-Difluoro benzoyl]Piperidine hydrochloride106266-04-0
179Risperidone
180Paliperidone3-(Benzyloxy)pyridine-2-amine24016-03-3
181Racecadotril2-Benzyl acrylic acid5669-19-2
182RacecadotrilBenzyl glycinate p-toluene sulfonate1738-76-7
183RipretinibPhenyl phenylcarbamate1106749
184RivaroxabanR)-4-chloro-N-(2-hydroxy-3-(4-(3-oxomorpholino)phenylamino)propyl)cyclopenta-1,3- dienecarboxamide.721401-53-2
185Rivaroxaban(S)-4-(4-(5-(aminomethyl)-2-oxooxazolidin-3-yl)phenyl)morpholin-3-one hydrochloride898543-06-1
186Sitagliptin1,2,4-Triazolo[4,3-a]pyrazine, 5,6,7,8-tetrahydro-3-(trifluoromethyl) hydrochloride762240-92-6
187Sitagliptin4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-one764667-65-4
188Sitagliptin(2Z)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazine-7(8H)-yl]-1-(2,4,5-trifluorophenyl)but-2-en-2-amine767340 -03 -4
189Solifenacin3-Quinuclidinone hydrochloride1193-65-3
190Tofacitinib4-chloro-7H-pyrrolo [2,3-d]pyrimidine3680-69-1
191Barcitinib
192Ruxolitinib
1931,4,7-TriMethyl-1,4,7-Triazacyclononane96556-05-7
194BOC-L-Glutamine13726-85-7
195(1-Methylpiperidin-4-Yl)Methanamine7149-42-0